SCHEMBL3797263

SCHEMBL3797263

CCOc1ncccc1C1(OC(=O)N2CCC(N3CCN(C)CC3)CC2)C(=O)N(S(=O)(=O)c2ccccc2OC)c2ccc(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 19/20 0.46
OXTR P30559 3/20 0.45
AVPR1A P37288 3/20 0.45
AVPR2 P30518 2/20 0.42
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
GPR65 Q8IYL9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794899 0.92 AVPR1B (0.43) AVPR1BOXTRAVPR1AAVPR2GPR65
SCHEMBL3803451 0.92 KDM4E (0.42) AVPR1BOXTRAVPR1A
SCHEMBL1591735 0.91 AVPR1B (0.54) AVPR1BOXTRAVPR1AAVPR2GPR65
SCHEMBL3797266 0.91 AVPR1B (0.46) AVPR1BOXTRAVPR1AAVPR2GPR65
SCHEMBL6526334 0.91 AVPR1B (0.51) AVPR1BOXTRAVPR1ACHRM2CHRM4
SCHEMBL1795556 0.90 AVPR1B (0.43) AVPR1BOXTRAVPR1AAVPR2GPR65
SCHEMBL27800666 0.89 KDM4E (0.41) AVPR1BOXTRAVPR1A
SCHEMBL15279969 0.88 ALDH1A1 (0.37) AVPR1BOXTRAVPR1AAVPR2CHRM2
SCHEMBL15279958 0.88 ALDH1A1 (0.37) AVPR1BOXTRAVPR1AAVPR2CHRM2
SCHEMBL6521609 0.88 AVPR1B (0.51) AVPR1BOXTRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231645-A2 5-HALOGEN-SUBSTITUTED OXINDOLE DERIVATIVES AND USE THEREOF FOR TREATING VASOPRESSINE-DEPENDENT DISEASES Abbott GmbH & Co. KG (DE) 2010-09-29 EP disclosed
WO-2009071689-A2 5-HALOGEN-SUBSTITUTED OXINDOLE DERIVATIVES AND USE THEREOF FOR TREATING VASOPRESSINE-DEPENDENT DISEASES ABBOTT GMBH & CO. KG (DE) 2009-06-11 WO disclosed