SCHEMBL3798481

SCHEMBL3798481

Cc1csc2ncnc(Nc3ccccc3OC3CCOCC3)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 7/20 0.47
MKNK1 Q9BUB5 5/20 0.47
SRC P12931 3/20 0.47
RAB9A P51151 2/20 0.43
LMNA P02545 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NOD2 Q9HC29 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.42
PIP4K2C Q8TBX8 1/20 0.42
MRGPRX1 Q96LB2 1/20 0.42
CDK2 P24941 1/20 0.41
FLT3 P36888 1/20 0.41
CCNA1 P78396 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.40
EGFR P00533 2/20 0.40
ERBB2 P04626 1/20 0.40
KDR P35968 2/20 0.39
KAT2B Q92831 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3795962 0.94 MKNK1 (0.44) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3795968 0.94 MKNK1 (0.44) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3797145 0.94 MKNK1 (0.44) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3799478 0.91 LMNA (0.45) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3803590 0.90 LMNA (0.45) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3796453 0.84 HSP90AB1 (0.43) MKNK2MKNK1RAB9ALMNARXFP1
SCHEMBL3805573 0.84 MKNK2 (0.55) MKNK2MKNK1SRCRAB9ALMNA
SCHEMBL3795880 0.84 MKNK2 (0.49) MKNK2MKNK1SRCEGFR
SCHEMBL3804308 0.83 MKNK2 (0.56) MKNK2MKNK1
SCHEMBL3801083 0.82 MKNK2 (0.50) MKNK2MKNK1RAB9ALMNARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100143341-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DEVELOGEN AKTIENGESELLSCHAFT (DE) 2010-06-10 US claimed
EP-1899353-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DeveloGen Aktiengesellschaft (DE) 2008-03-19 EP claimed
WO-2007059905-A9 THIENOPYRIMIDINES TREATING INFLAMMATORY DISEASES DEVELOGEN AG (DE) 2007-11-01 WO claimed
WO-2007059905-A2 THIENOPYRIMIDINES TREATING INFLAMMATORY DISEASES DEVELOGEN AKTIENGESELLSCHAFT (DE) 2007-05-31 WO claimed
WO-2006136402-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DEVELOGEN AKTIENGESELLSCHAFT (DE) 2006-12-28 WO claimed
US-20100143341-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DEVELOGEN AKTIENGESELLSCHAFT (DE) 2010-06-10 US disclosed
EP-1899353-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DeveloGen Aktiengesellschaft (DE) 2008-03-19 EP disclosed
WO-2007059905-A9 THIENOPYRIMIDINES TREATING INFLAMMATORY DISEASES DEVELOGEN AG (DE) 2007-11-01 WO disclosed
WO-2007059905-A2 THIENOPYRIMIDINES TREATING INFLAMMATORY DISEASES DEVELOGEN AKTIENGESELLSCHAFT (DE) 2007-05-31 WO disclosed
WO-2006136402-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DEVELOGEN AKTIENGESELLSCHAFT (DE) 2006-12-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100143341-A1 THIENOPYRIMIDINES FOR PHARMACEUTICAL COMPOSITIONS DTYMK, CMPK1, PDXK MKNK2 21/4885MKNK1 74/4885SRC 1573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.