SCHEMBL3799197

SCHEMBL3799197

CN(Cc1cc(-c2ccccc2Br)c(S(=O)(=O)c2cccnc2)s1)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.35
NAMPT P43490 2/20 0.34
F2 P00734 2/20 0.34
GLS O94925 1/20 0.34
PTGER2 P43116 6/20 0.34
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
ALPL P05186 1/20 0.32
TACR1 P25103 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
CLK1 P49759 1/20 0.31
AGTR2 P50052 1/20 0.31
RIPK1 Q13546 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654305 0.93 GPBAR1 (0.35) SOS1NAMPTF2GLSPTGER2
SCHEMBL4132659 0.87 NAMPT (0.39) NAMPTPTGER2
SCHEMBL3648432 0.87 GPBAR1 (0.39) NAMPTF2PTGER2HTR2CSLC6A4
SCHEMBL3649650 0.83 NAMPT (0.36) SOS1NAMPTF2GLSPTGER2
SCHEMBL3799201 0.82 PTGER2 (0.35) NAMPTPTGER2ABCC9ABCC8KCNJ11
SCHEMBL3650554 0.81 HTR2C (0.37) SOS1NAMPTF2GLSHTR2C
SCHEMBL3654644 0.79 HTR2C (0.38) SOS1F2GLSHTR2CSLC6A4
SCHEMBL3654491 0.79 NAMPT (0.35) SOS1NAMPTF2GLSPTGER2
SCHEMBL3654948 0.79 F2 (0.35) SOS1F2GLSHTR2CSLC6A4
Carbamic Acid SCHEMBL3651234 0.79 HTR2C (0.37) SOS1F2GLSHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed