SCHEMBL3648432

SCHEMBL3648432

CN(Cc1cc(-c2cccnc2Cl)c(S(=O)(=O)c2cccnc2)s1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.39
F2 P00734 3/20 0.34
RXFP1 Q9HBX9 1/20 0.33
PTGER2 P43116 6/20 0.33
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 1/20 0.32
ALOX12 P18054 1/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
NAMPT P43490 1/20 0.32
AGTR2 P50052 1/20 0.32
ABCC9 O60706 1/20 0.31
ABCC8 Q09428 1/20 0.31
KCNJ11 Q14654 1/20 0.31
KCNJ8 Q15842 1/20 0.31
CLK1 P49759 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3650554 0.92 HTR2C (0.37) GPBAR1F2RXFP1HTR2CSLC6A4
SCHEMBL3645987 0.88 GPBAR1 (0.36) GPBAR1F2RXFP1PTGER2HTR2C
SCHEMBL4130745 0.88 GPBAR1 (0.40) GPBAR1RXFP1PTGER2ALDH1A1PKM
SCHEMBL3799197 0.87 SOS1 (0.35) F2PTGER2HTR2CSLC6A4NAMPT
Hydrochloric Acid SCHEMBL3654116 0.84 HTR6 (0.35) GPBAR1F2RXFP1PTGER2ALDH1A1
SCHEMBL3803075 0.83 ALDH1A1 (0.33) GPBAR1F2ALDH1A1HTR2CSLC6A4
SCHEMBL3648440 0.82 GPBAR1 (0.38) GPBAR1RXFP1PTGER2NAMPTABCC9
SCHEMBL3654948 0.82 F2 (0.35) GPBAR1F2HTR2CSLC6A4AGTR2
SCHEMBL3654305 0.81 GPBAR1 (0.35) GPBAR1F2PTGER2NAMPT
SCHEMBL3651630 0.81 HTR2C (0.32) HTR2CSLC6A4AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed