SCHEMBL3799201

SCHEMBL3799201

CC(C)(C)CN(Cc1cc(-c2ccccc2Br)c(S(=O)(=O)c2cccnc2)s1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGER2 P43116 6/20 0.35
NAMPT P43490 6/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
KCNA5 P22460 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 3/20 0.32
TP53 P04637 2/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654310 0.93 GPBAR1 (0.34) PTGER2NAMPT
SCHEMBL3648440 0.87 GPBAR1 (0.38) PTGER2NAMPTMAPTLMNATP53
SCHEMBL4132659 0.86 NAMPT (0.39) PTGER2NAMPTKDM4EMAPTKCNA5
SCHEMBL3649653 0.82 PTGER2 (0.39) PTGER2NAMPTKMT2ALMNATP53
SCHEMBL3799197 0.82 SOS1 (0.35) PTGER2NAMPTABCC9ABCC8KCNJ11
SCHEMBL3650557 0.81 GPBAR1 (0.35) NAMPTKDM4EKMT2A
SCHEMBL3654647 0.80 CNR2 (0.35) KDM4EMAPTKMT2ALMNA
Carbamic Acid SCHEMBL3651238 0.79 CA12 (0.33) KDM4EMAPTKMT2ALMNA
SCHEMBL3652839 0.79 CTSK (0.32) NAMPT
SCHEMBL3654497 0.79 GPBAR1 (0.36) PTGER2NAMPTKMT2ALMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed