SCHEMBL3801726

SCHEMBL3801726

CC(C)CCOc1cc(-c2cn[nH]c2)ccc1N

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.69
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TLR8 Q9NR97 1/20 0.41
MELK Q14680 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
ROCK1 Q13464 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621595 0.86 ALDH1A1 (0.59) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3801724 0.82 HTT (0.54) ROCK2MELKROCK1LRRK2
SCHEMBL3713992 0.82 ROCK2 (1.00) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3656438 0.77 ALDH1A1 (0.67) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3718200 0.76 ROCK2 (0.61) ROCK2HSD17B10ROCK1
SCHEMBL3714540 0.75 ROCK2 (0.60) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3722814 0.75 ROCK2 (0.60) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3808767 0.74 ROCK2 (0.58) ROCK2KDM4EMEN1ALDH1A1POLB
SCHEMBL3714084 0.74 ROCK2 (0.71) ROCK2MELKROCK1
SCHEMBL3810004 0.74 GSK3B (0.38) ROCK2MAPTKMT2ATLR8GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed