Iotroxic Acid

Iotroxic Acid

SCHEMBL38038

O=C(COCCOCCOCC(=O)Nc1c(I)cc(I)c(C(=O)O)c1I)Nc1c(I)cc(I)c(C(=O)O)c1I

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.65
MAPK1 P28482 1/20 0.65
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.31
HIF1A Q16665 1/20 0.30
EPAS1 Q99814 1/20 0.30
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iotetric Acid SCHEMBL37863 1.00 TSHR (0.65) TSHRMAPK1KDM4ENPC1MAPT
Iotetric Acid SCHEMBL27748028 1.00 TSHR (0.65) TSHRMAPK1KDM4ENPC1MAPT
Iotroxic Acid SCHEMBL27729545 1.00 TSHR (0.65) TSHRMAPK1KDM4ENPC1MAPT
Iotrizoic Acid SCHEMBL31409209 0.94 TSHR (0.58) TSHRMAPK1KDM4ENPC1MAPT
Iotrizoic Acid SCHEMBL2111608 0.94 TSHR (0.58) TSHRMAPK1KDM4ENPC1MAPT
Ioglycamic Acid SCHEMBL29881458 0.93 TSHR (0.70) TSHRMAPK1KDM4ENPC1MAPT
Ioglycamic Acid SCHEMBL433485 0.93 TSHR (0.70) TSHRMAPK1KDM4ENPC1MAPT
Iodoxamic Acid SCHEMBL377402 0.89 TSHR (0.74) TSHRMAPK1NPC1RAB9APOLB
SCHEMBL12142383 0.89 TSHR (0.74) TSHRMAPK1NPC1RAB9APOLB
Iodoxamic Acid SCHEMBL29397252 0.89 TSHR (0.74) TSHRMAPK1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1197 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021238893-A1 EFFICIENT AND EFFECTIVE TISSUE CLEARING AGENTS AND THEIR COMPOSITIONS THE CHINESE UNIVERSITY OF HONG KONG (CN) 2021-12-02 WO claimed
US-20170066828-A1 Humanized Anti-HLA-DR Antibodies IMMUNOMEDICS, INC. 2017-03-09 US claimed
US-20160375234-A1 TRANSPAPILLARY METHODS AND COMPOSITIONS FOR DIAGNOSING AND TREATING BREAST CONDITIONS ATOSSA THERAPEUTICS, INC. 2016-12-29 US claimed
EP-3092027-A1 TRANSPAPILLARY METHODS AND COMPOSITIONS FOR DIAGNOSING AND TREATING BREAST CONDITIONS Atossa Genetics Inc. (US) 2016-11-16 EP claimed
US-9393325-B2 Bioabsorbable co-filler for cerebrovascular aneurysms ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2016-07-19 US claimed
US-20160151124-A1 IMPLANTABLE MARKERS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2016-06-02 US claimed
EP-3019208-A1 IMPLANTABLE MARKERS Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2016-05-18 EP claimed
EP-1521775-B1 MONOCLONAL ANTIBODY PAM4 AND ITS USE FOR DIAGNOSIS AND THERAPY OF PANCREATIC CANCER IMMUNOMEDICS INC (US) 2015-09-09 EP claimed
WO-2015106094-A1 TRANSPAPILLARY METHODS AND COMPOSITIONS FOR DIAGNOSING AND TREATING BREAST CONDITIONS Atossa Genetics Inc. (US) 2015-07-16 WO claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
EP-0703790-B1 IODINATED PARAMAGNETIC CHELATES, AND THEIR USE AS CONTRAST AGENTS BRACCO SPA (IT) 2000-08-16 EP claimed
EP-0576740-B1 Process and device for the preparation of a contrast medium from a concentrate SCHERING AG (DE) 1998-07-29 EP claimed
US-5662930-A SURFACE MODIFICATION THE LIPOSOME COMPANY, INC. (US) 1997-09-02 US claimed
US-5660814-A Iodinated paramagnetic chelates, and their use as contrast agents DIBRA S.P.A. (IT) 1997-08-26 US claimed
US-5614214-A INCORPORATING LIPID, REDUCING BLOOD PRESSURE DECREASE THE LIPOSOME COMPANY, INC. (US) 1997-03-25 US claimed
EP-0703790-A1 IODINATED PARAMAGNETIC CHELATES, AND THEIR USE AS CONTRAST AGENTS BRACCO S.p.A. (IT) 1996-04-03 EP claimed
EP-0699068-A1 REDUCTION OF LIPOSOME-INDUCED ADVERSE PHYSIOLOGICAL REACTIONS THE LIPOSOME COMPANY, INC. (US) 1996-03-06 EP claimed
US-5450847-A Process for making doses formulation of contrast media from concentrate SCHERING AKTIENGESELLSCHAFT (DE) 1995-09-19 US claimed
WO-1994027644-A1 IODINATED PARAMAGNETIC CHELATES, AND THEIR USE AS CONTRAST AGENTS BRACCO S.P.A. (IT) 1994-12-08 WO claimed
WO-1994027580-A1 REDUCTION OF LIPOSOME-INDUCED ADVERSE PHYSIOLOGICAL REACTIONS THE LIPOSOME COMPANY, INC. (US) 1994-12-08 WO claimed