SCHEMBL3811441

SCHEMBL3811441

CC(=O)Nc1ccc2c(c1)CCC(I)C2=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.59
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
MAOA P21397 2/20 0.50
CYP1A2 P05177 1/20 0.50
ADRA2A P08913 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR2C P28335 1/20 0.50
SLC6A4 P31645 1/20 0.50
HTR2B P41595 1/20 0.50
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trimethylammonium SCHEMBL10341484 0.96 BAZ2B (0.56) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL4579245 0.85 BAZ2B (0.55) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL10908114 0.84 BAZ2B (0.58) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL7653688 0.81 BAZ2B (0.54) BAZ2BNPC1RAB9AMAOACYP1A2
Iodide SCHEMBL10341485 0.81 BAZ2B (0.54) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL6792959 0.81 BAZ2B (0.54) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL5582823 0.80 ITGB3 (0.66) BAZ2BNPC1RAB9AMTNR1AITGB3
SCHEMBL5582711 0.79 BAZ2B (0.52) BAZ2BNPC1RAB9AMTNR1AITGB3
SCHEMBL29113471 0.79 BAZ2B (0.52) BAZ2BNPC1RAB9AMAOACYP1A2
SCHEMBL10341502 0.79 ITGB3 (0.59) BAZ2BNPC1RAB9AMAOACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2089367-A1 PYRAZOLINE COMPOUNDS AS MINERALOCORTICOID RECEPTOR ANTAGONISTS Pfizer Products Incorporated (US) 2009-08-19 EP disclosed
WO-2008053300-A1 PYRAZOLINE COMPOUNDS AS MINERALOCORTICOID RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 2008-05-08 WO disclosed