Clarithromycin

Clarithromycin

SCHEMBL38124

CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)C(C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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The experimentally established mechanism targets of Clarithromycin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 1.00
KCNH2 Q12809 5/20 1.00
ABCB1 P08183 2/20 1.00
SLCO1B3 Q9NPD5 2/20 1.00
SLCO1B1 Q9Y6L6 2/20 1.00
AR P10275 1/20 1.00
MAPK1 P28482 1/20 1.00
MLNR O43193 2/20 0.92
TSHR P16473 2/20 0.92
LMNA P02545 2/20 0.92
TDP1 Q9NUW8 1/20 0.92
ALB P02768 1/20 0.92
CNR1 P21554 1/20 0.92
HTR2A P28223 1/20 0.92
AOX1 Q06278 1/20 0.92
CYP1B1 Q16678 1/20 0.92
ABCC4 O15439 1/20 0.77
ABCB11 O95342 1/20 0.77
PGR P06401 1/20 0.77
HTR1A P08908 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clarithromycin SCHEMBL13210325 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL15472892 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL1176361 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL38125 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL24064961 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL17705916 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL23309064 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL14010008 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL23854898 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1
Clarithromycin SCHEMBL12296733 1.00 CYP3A4 (1.00) CYP3A4KCNH2ABCB1SLCO1B3SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 65506 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
US-20260138957-A1 UREA-LINKED 2-AMINOIMIDAZOLE DIMER POTENTIATORS UNIVERSITY OF NOTRE DAME DU LAC (US) 2026-05-21 US claimed
WO-2026107208-A1 COMPOSITIONS AND METHODS FOR TREATING MICROBIAL INFECTIONS THE METHODIST HOSPITAL (US) 2026-05-21 WO claimed
EP-4744729-A2 METHODS OF TREATING GASTROINTESTINAL STROMAL TUMORS Deciphera Pharmaceuticals, LLC (US) 2026-05-20 EP claimed
EP-4007582-B1 ANTIBIOTICS IN COMBINATION WITH PHOTODYNAMIC THERAPY FOR USE IN A METHOD OF ENHANCING THE ANTIMICROBIAL ACTION OF SYSTEMICALLY ADMINISTERED ANTIBIOTICS KOITE HEALTH OY (FI) 2026-05-20 EP claimed
US-12629363-B2 Prophylaxis and treatment of angioedema PHARVARIS GMBH (CH) 2026-05-19 US claimed
CN-122056853-A Antibacterial agent based on graphite phase carbon nitride, and preparation method and application thereof 海南医科大学(海南省医学科学院) 2026-05-19 CN claimed
WO-2026102345-A1 METHODS OF ADMINISTERING THE VOLTAGE-GATED POTASSIUM CHANNEL OPENER AZETUKALNER XENON PHARMACEUTICALS INC. (CA) 2026-05-15 WO claimed
CN-122042848-A Method for separating and measuring key starting materials and related compounds of clavulanone by HPLC (high Performance liquid chromatography) 福建大谱生物医药有限公司 2026-05-15 CN claimed
US-4921839-A Erythromycin a 11,12-carbonate 9-oxime derivatives BEECHAM GROUP P.L.C. (GB) 1990-05-01 US claimed
EP-0180415-B1 A 6-0-methylerythromycin A derivative TAISHO PHARMACEUTICAL CO. LTD (JP) 1990-01-31 EP claimed
US-4808411-A ERYTHROMYCIN AND CARBOMER ABBOTT LABORATORIES (US) 1989-02-28 US claimed
EP-0195960-B1 METHOD FOR SELECTIVE METHYLATION OF ERYTHROMYCIN A DERIVATIVES TAISHO PHARMACEUTICAL CO. LTD (JP) 1988-12-14 EP claimed
EP-0293885-A2 Antibiotic-polymer compositions ABBOTT LABORATORIES (US) 1988-12-07 EP claimed
EP-0260938-A2 Erythromycin A derivatives and method for preparing the same TAISHO PHARMACEUTICAL CO. LTD (JP) 1988-03-23 EP claimed
EP-0245012-A1 Method for the preparation of 14-hydroxy-6-0-methyl-erythromycin A TAISHO PHARMACEUTICAL CO. LTD (JP) 1987-11-11 EP claimed
US-4680386-A 6-O-methylerythromycin a derivative TAISHO PHARMACEUTICAL CO., LTD. (JP) 1987-07-14 US claimed
EP-0194833-A2 Erythromycin derivatives BEECHAM GROUP PLC (GB) 1986-09-17 EP claimed
EP-0180415-A2 A 6-0-methylerythromycin A derivative TAISHO PHARMACEUTICAL CO. LTD (JP) 1986-05-07 EP claimed