SCHEMBL3815467

SCHEMBL3815467

FC(F)(F)Oc1cccc2c1C=CNC2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
KDM4E B2RXH2 1/20 0.33
GRIA1 P42261 3/20 0.32
CACNG8 Q8WXS5 3/20 0.32
CCR3 P51677 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
CACNG2 Q9Y698 1/20 0.30
PNMT P11086 1/20 0.30
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4727743 0.78 PARP1 (0.43) PARP1PNMT
SCHEMBL31158971 0.69 CD44 (0.37) KDM4EGRIA1CACNG8HTR2AHTR2C
SCHEMBL31176882 0.69 POLB (0.40) PARP1
SCHEMBL28067181 0.68 PARP1 (0.47) PARP1HTR2CHTR2BPNMT
SCHEMBL13833540 0.68 PARP1 (0.47) PARP1HTR2C
SCHEMBL14820465 0.68 PARP1 (0.47) PARP1
SCHEMBL16621278 0.68 PARP1 (0.47) PARP1PNMT
SCHEMBL16154709 0.68 PARP1 (0.43) PARP1
SCHEMBL28039591 0.67 SRC (0.44) PARP1KDM4EGRIA1CACNG8CCR3
SCHEMBL28122218 0.66 PDE3A (0.34) PARP1GRIA1CACNG8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1684787-A4 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2009-08-05 EP disclosed
EP-1684787-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2006-08-02 EP disclosed
WO-2005051410-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-06-09 WO disclosed