SCHEMBL3818896

SCHEMBL3818896

COc1cnc2cccc([C@@H](CNC(=O)OC(C)(C)C)C3CCC(=O)CC3)c2n1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 2/20 0.34
ACACB O00763 5/20 0.34
ACACA Q13085 3/20 0.34
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
CKS1B P61024 2/20 0.33
SKP1 P63208 2/20 0.33
SKP2 Q13309 2/20 0.33
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
GFER P55789 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BCHE P06276 1/20 0.32
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
PCSK9 Q8NBP7 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3888157 0.90 ACACB (0.34) CPB2ACACBACACAKDM4ETDP1
SCHEMBL1711909 0.81 KDM4E (0.38) KDM4ETDP1GFERHSD17B10L3MBTL1
SCHEMBL1712711 0.81 KDM4E (0.38) KDM4ETDP1GFERHSD17B10L3MBTL1
SCHEMBL2539541 0.80 SCN9A (0.36) KDM4EMTNR1AMTNR1BALDH1A1
SCHEMBL2539534 0.80 SCN9A (0.36) KDM4EMTNR1AMTNR1BALDH1A1
SCHEMBL1711958 0.80 MTNR1B (0.39) KDM4ETDP1GFERHSD17B10L3MBTL1
SCHEMBL2286483 0.80 MTNR1B (0.39) KDM4ETDP1CKS1BSKP1SKP2
SCHEMBL3819813 0.78
SCHEMBL1711908 0.74 KDM4E (0.39) KDM4ETDP1MTNR1AMTNR1BALDH1A1
SCHEMBL1712708 0.74 KDM4E (0.39) KDM4ETDP1MTNR1AMTNR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094267-B1 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2015-04-22 EP disclosed
EP-2094267-A2 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-09-02 EP disclosed
WO-2008078305-A2 4-(1-AMINO-ETHYL)-CYCLOHEXYLAMINE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-03 WO disclosed