SCHEMBL3820120

SCHEMBL3820120

CCN(c1nc(CN(c2ccc(F)cc2)[C@H](CC(C)C)C(N)=O)cs1)C1CC1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.33
CNR2 P34972 3/20 0.32
CNR1 P21554 2/20 0.32
BCHE P06276 4/20 0.32
GRIA2 P42262 5/20 0.31
GRIN2A Q12879 5/20 0.31
HCRTR1 O43613 1/20 0.31
S1PR1 P21453 1/20 0.31
GRIN1 Q05586 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3816257 1.00 CAPN1 (0.33) CAPN1CNR2CNR1BCHEGRIA2
SCHEMBL3816035 0.87 ITGB3 (0.35)
SCHEMBL3822022 0.83 PTGDR2 (0.38) CAPN1CNR2CNR1BCHE
SCHEMBL3820116 0.83 CAPN1 (0.34) CAPN1BCHEGRIA2GRIN2AHCRTR1
SCHEMBL3816250 0.83 CAPN1 (0.34) CAPN1BCHEGRIA2GRIN2AHCRTR1
SCHEMBL3821711 0.81 DPP4 (0.37) BCHE
SCHEMBL8187785 0.80 GRM1 (0.33) CAPN1BCHEGRIA2GRIN2AHCRTR1
SCHEMBL3822210 0.80 GRIN2A (0.39) GRIA2GRIN2AGRIN1
SCHEMBL3821866 0.80 S1PR1 (0.38) CNR2CNR1S1PR1
SCHEMBL3822208 0.79 GRM1 (0.34) GRIA2GRIN2AHCRTR1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091917-A1 ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2009-08-26 EP claimed
WO-2008073934-A1 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed