SCHEMBL3820149

SCHEMBL3820149

CN(CCC(=O)Cl)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
ALDH1A1 P00352 3/20 0.39
TP53 P04637 1/20 0.39
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.31
PHF8 Q9UPP1 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3824058 0.86 ALDH1A1 (0.46) TSHRALDH1A1TP53NPC1RAB9A
SCHEMBL3821521 0.84 ALDH1A1 (0.46) TSHRALDH1A1TP53PHF8KDM2A
SCHEMBL3823996 0.82 ALDH1A1 (0.50) TSHRALDH1A1TP53PHF8KDM2A
SCHEMBL1869025 0.79 PHF8 (0.46) ALDH1A1PHF8KDM2A
SCHEMBL3763074 0.78 NPC1 (0.36) TSHRALDH1A1NPC1RAB9AKMT2A
SCHEMBL19133282 0.77 ALDH1A1 (0.45) ALDH1A1NPC1RAB9AKMT2APHF8
SCHEMBL19924618 0.77 ALDH1A1 (0.43) TSHRALDH1A1NPC1RAB9A
SCHEMBL4034999 0.76 ALDH1A1 (0.34) ALDH1A1NPC1RAB9A
SCHEMBL645133 0.76
SCHEMBL3297922 0.75 ALDH1A1 (0.46) ALDH1A1NPC1RAB9AKMT2APHF8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987026-B1 AMINOACYL PRODRUG DERIVATIVES AND MEDICAMENTS FOR THE TREATMENT OF THROMBOEMBOLITIC DISORDERS BAYER HEALTHCARE AG (DE) 2009-08-26 EP disclosed
EP-1987026-A1 AMINOACYL PRODRUG DERIVATIVES AND MEDICAMENTS FOR THE TREATMENT OF THROMBOEMBOLITIC DISORDERS Bayer HealthCare AG (DE) 2008-11-05 EP disclosed
WO-2007093328-A1 AMINOACYL PRODRUG DERIVATIVES AND MEDICAMENTS FOR THE TREATMENT OF THROMBOEMBOLITIC DISORDERS BAYER HEALTHCARE AG (DE) 2007-08-23 WO disclosed