SCHEMBL38205

SCHEMBL38205

Cc1c(C(=O)O)sc2c(=O)[nH]c(Cc3cccc(Cl)c3)nc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.64
PDE9A O76083 1/20 0.52
PDE1A P54750 1/20 0.52
PDE1B Q01064 1/20 0.52
PDE1C Q14123 1/20 0.52
PIM1 P11309 6/20 0.44
PIM2 Q9P1W9 4/20 0.43
PIM3 Q86V86 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
RNASEH1 O60930 1/20 0.41
CCNB2 O95067 1/20 0.41
CCNE2 O96020 1/20 0.41
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3492352 0.84 PDE5A (0.69) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL3492211 0.83 PDE5A (0.67) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL37798 0.78 PDE5A (1.00) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL3493794 0.77 KMT2A (0.59) PDE5AKDM4EALDH1A1KMT2A
SCHEMBL401142 0.76 PDE5A (0.64) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL37776 0.74 PDE5A (0.61) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL3492301 0.74 PDE5A (1.00) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL16175769 0.74 PDE5A (0.63) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL3492213 0.74 PDE5A (0.60) PDE5APDE9APDE1APDE1BPDE1C
SCHEMBL37864 0.73 PDE5A (0.82) PDE5APDE9APDE1APDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed