SCHEMBL3821499

SCHEMBL3821499

COC(=O)OC1CCN(c2ccc(F)c(C)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACACB O00763 9/20 0.46
PTGES O14684 1/20 0.40
HRH3 Q9Y5N1 5/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
USP30 Q70CQ3 1/20 0.39
DRD4 P21917 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3820953 0.87 NOTUM (0.41) ACACBPTGESHRH3ALDH1A1MAPT
SCHEMBL5481745 0.82 MAPT (0.55) PTGESALDH1A1MAPT
SCHEMBL31381229 0.77 NOTUM (0.56) PTGES
SCHEMBL3820949 0.77 NOTUM (0.56) PTGES
SCHEMBL8127380 0.76 ADRB1 (0.41) PTGESALDH1A1
SCHEMBL31381251 0.76 PDK2 (0.49) PTGESALDH1A1MAPT
SCHEMBL6206254 0.72 ALDH1A1 (0.51) ALDH1A1MAPT
SCHEMBL13723405 0.71 NOTUM (0.44) PTGESALDH1A1
SCHEMBL29621605 0.71 NOTUM (0.53) PTGES
SCHEMBL28747907 0.71 MAPT (0.50) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685123-B1 SUBSTITUTED DIHYDROQUINAZOLINES II BAYER HEALTHCARE AG (DE) 2009-08-19 EP disclosed
EP-1685123-A2 SUBSTITUTED DIHYDROQUINAZOLINES II Bayer HealthCare AG (DE) 2006-08-02 EP disclosed
WO-2005047278-A2 SUBSTITUTED DIHYDROQUINAZOLINES II BAYER HEALTHCARE AG (DE) 2005-05-26 WO disclosed