SCHEMBL382255

SCHEMBL382255

CCOC(=O)c1ccc(N2CCN(Cc3nc4ccccc4[nH]3)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.66
GAA P10253 1/20 0.66
DRD4 P21917 17/20 0.66
HTR1A P08908 1/20 0.62
ADRA2C P18825 1/20 0.62
HTR2A P28223 1/20 0.62
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
MAPT P10636 1/20 0.59
MAPK1 P28482 1/20 0.59
RAB9A P51151 1/20 0.59
DRD2 P14416 4/20 0.54
DRD3 P35462 1/20 0.53
HPGD P15428 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652040 0.85 MAPT (0.57) NPC1GAAALDH1A1LMNAMAPT
SCHEMBL383213 0.85 DRD4 (0.77) NPC1GAADRD4HTR1AADRA2C
SCHEMBL9543721 0.82 DRD4 (0.59) NPC1GAADRD4HTR1AADRA2C
SCHEMBL4814328 0.80 NPC1 (1.00) NPC1GAADRD4HTR1AADRA2C
SCHEMBL4809921 0.80 DRD4 (1.00) NPC1GAADRD4HTR1AADRA2C
SCHEMBL8689422 0.79 DRD4 (1.00) NPC1GAADRD4HTR1AADRA2C
SCHEMBL9302827 0.78 MAPT (0.71) NPC1GAAALDH1A1LMNAMAPT
SCHEMBL8687797 0.78 DRD4 (1.00) NPC1GAADRD4HTR1AADRA2C
SCHEMBL6787298 0.78 DRD4 (1.00) NPC1GAADRD4HTR1AADRA2C
SCHEMBL3318522 0.78 PRMT1 (0.68) DRD4HTR2AALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US disclosed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP disclosed