SCHEMBL383213

SCHEMBL383213

O=C(O)c1ccc(N2CCN(Cc3nc4ccccc4[nH]3)CC2)cc1

nearest known ligand 0.77

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 16/20 0.77
NPC1 O15118 1/20 0.74
GAA P10253 1/20 0.74
HTR1A P08908 1/20 0.64
ADRA2C P18825 1/20 0.64
HTR2A P28223 1/20 0.64
DRD2 P14416 3/20 0.61
DRD3 P35462 1/20 0.61
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
CYP3A4 P08684 1/20 0.57
ALOX15 P16050 1/20 0.57
OPRK1 P41145 1/20 0.57
SIGMAR1 Q99720 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4809921 0.88 DRD4 (1.00) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL4814328 0.85 NPC1 (1.00) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL382255 0.85 NPC1 (0.66) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL8687797 0.83 DRD4 (1.00) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL6787298 0.83 DRD4 (1.00) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL23964171 0.82 DRD4 (0.82) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL7651404 0.82 HTR2B (0.65) HPGDKDM4EALDH1A1
SCHEMBL5157052 0.81 HTT (0.84) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL31267420 0.81 DRD4 (0.72) DRD4NPC1GAAHTR1AADRA2C
SCHEMBL16795300 0.80 DRD4 (0.67) DRD4NPC1GAADRD2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US disclosed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP disclosed