SCHEMBL3827262

SCHEMBL3827262

C#Cc1cnc2c(c1)c(O)c(C(=O)NCC(=O)OCCCC)c(=O)n2C

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
EGLN1 Q9GZT9 3/20 0.39
POLB P06746 1/20 0.38
HIF1A Q16665 15/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828180 0.86 ATM (0.43) ATML3MBTL1EGLN1POLBHIF1A
SCHEMBL2579371 0.85 EGLN1 (0.41) EGLN1HIF1A
SCHEMBL2582355 0.84 EGLN1 (0.52) EGLN1HIF1A
SCHEMBL2579364 0.75 EGLN1 (0.41) EGLN1HIF1A
SCHEMBL12101566 0.75 L3MBTL1 (0.41) L3MBTL1EGLN1POLBHIF1A
SCHEMBL2583556 0.75 EGLN1 (0.45) EGLN1HIF1A
SCHEMBL2581713 0.74 EGLN1 (0.52) EGLN1HIF1A
SCHEMBL2580152 0.74 GABRA1 (0.41) EGLN1HIF1A
SCHEMBL2583492 0.73 EGLN1 (0.55) EGLN1HIF1A
SCHEMBL2578789 0.73 EGLN1 (0.57) EGLN1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097416-A1 AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF Amgen, Inc (US) 2009-09-09 EP disclosed
WO-2008076425-A1 AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF AMGEN INC. (US) 2008-06-26 WO disclosed