SCHEMBL3828084

SCHEMBL3828084

NNC(=O)c1ccc(Sc2cccc(OCc3ccccc3)c2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
S1PR1 P21453 1/20 0.53
ALDH1A1 P00352 3/20 0.53
SMPD1 P17405 1/20 0.47
MAPT P10636 1/20 0.47
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
NR4A2 P43354 1/20 0.45
SPHK2 Q9NRA0 4/20 0.45
SIRT2 Q8IXJ6 1/20 0.44
SPHK1 Q9NYA1 2/20 0.44
MAOB P27338 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4408927 0.86 MAOB (0.56) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL28125444 0.85 S1PR1 (0.51) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL13596044 0.84 MAPT (0.65) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL3844659 0.80 MAOB (0.52) RAB9ASMN1; SMN2S1PR1MAPTNR4A2
SCHEMBL3825466 0.79 DHODH (0.47) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6031320 0.77 KDM4E (0.57) S1PR1ALDH1A1SMPD1NR4A2MAOB
SCHEMBL6031317 0.77 KDM4E (0.57) S1PR1ALDH1A1SMPD1NR4A2MAOB
SCHEMBL3085911 0.77 MAOB (0.52) NPC1RAB9AS1PR1ALDH1A1NR4A2
SCHEMBL14295927 0.77 S1PR1 (0.48) SMN1; SMN2MEN1KMT2AS1PR1SMPD1
SCHEMBL3832329 0.76 ALDH1A1 (0.43) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090318389-A1 AGONISTS OF THE SPHINGOSINE-1 PHOSPHATE RECEPTOR PRAECIS PHARMACEUTICALS INCORPORATED (US) 2009-12-24 US disclosed
US-20090318389-A1 AGONISTS OF THE SPHINGOSINE-1 PHOSPHATE RECEPTOR PRAECIS PHARMACEUTICALS INCORPORATED (US) 2009-12-24 US disclosed
US-20090318389-A1 AGONISTS OF THE SPHINGOSINE-1 PHOSPHATE RECEPTOR PRAECIS PHARMACEUTICALS INCORPORATED (US) 2009-12-24 US disclosed
EP-2099768-A2 AGONISTS OF THE SPHINGOSINE-1-PHOSPHATE RECEPTOR Praecis Pharmaceuticals Incorporated (US) 2009-09-16 EP disclosed
WO-2008019090-A2 AGONISTS OF THE SPHINGOSINE-1-PHOSPHATE RECEPTOR PRAECIS PHARMACEUTICALS INCORPORATED (US) 2008-02-14 WO disclosed
WO-2008019090-A2 AGONISTS OF THE SPHINGOSINE-1-PHOSPHATE RECEPTOR PRAECIS PHARMACEUTICALS INCORPORATED (US) 2008-02-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318389-A1 AGONISTS OF THE SPHINGOSINE-1 PHOSPHATE RECEPTOR S1PR1, S1PR3, S1PR5 NPC1 1484/4885RAB9A 1514/4885SMN1; SMN2 1622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.