SCHEMBL3828550

SCHEMBL3828550

COCCN(CCOC)N(C)c1ccc(C(=O)C(=O)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.54
HPGD P15428 4/20 0.52
CES2 O00748 9/20 0.46
CES1 P23141 8/20 0.46
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
EGFR P00533 2/20 0.40
MAPT P10636 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828647 0.80 RAB9A (0.62) RAB9AHPGDCES2CES1NPC1
SCHEMBL3829873 0.76 RAB9A (0.71) RAB9AHPGDCES2CES1NPC1
Benzil SCHEMBL27731550 0.72 HPGD (0.62) RAB9AHPGDCES2CES1
SCHEMBL4140401 0.71 RAB9A (1.00) RAB9AHPGDCES2CES1NPC1
SCHEMBL634452 0.71 NAMPT (0.56) RAB9AHDAC1HDAC6KMT2A
SCHEMBL1756743 0.70 MEN1 (0.45) RAB9AHPGDNPC1ALDH1A1HTT
SCHEMBL30671562 0.70 RAB9A (0.96) RAB9AHPGDCES2CES1NPC1
Benzil SCHEMBL27395782 0.69 CES2 (0.64) RAB9AHPGDCES2CES1ALDH1A1
SCHEMBL22077519 0.69 NAMPT (0.56) HPGDALDH1A1MAPTHDAC1HDAC6
SCHEMBL29992460 0.69 MAPK1 (0.49) HDAC1HDAC6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0999835-B1 IMIDAZOLE DERIVATIVES AS MDR MODULATORS TAIJI BIOMEDICAL INC (US) 2009-09-09 EP disclosed
US-5840721-A INCREASE SENSITIVITY OF MULTIDRUG RESISTANT TUMOR CELLS TO ANTICANCER AGENTS ONTOGEN CORPORATION (US) 1998-11-24 US disclosed