SCHEMBL3828801

SCHEMBL3828801

CCOC(=O)c1c[nH]nc1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
MAPT P10636 4/20 0.45
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 1/20 0.44
JAK2 O60674 2/20 0.43
JAK3 P52333 2/20 0.43
KDM4E B2RXH2 2/20 0.42
RAB9A P51151 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41
HPGD P15428 1/20 0.41
POLB P06746 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13374014 0.79 KMT2A (0.46) TSHRMAPTALDH1A1HSD17B10KDM4E
SCHEMBL69229 0.78 KDM4E (0.54) TSHRMAPTALDH1A1KDM4ENPSR1
SCHEMBL5306579 0.77 TSHR (0.46) TSHRMAPTALDH1A1HSD17B10JAK2
SCHEMBL5778710 0.76 SMN1; SMN2 (0.52) TSHRMAPTALDH1A1HSD17B10KDM4E
SCHEMBL2921221 0.75 JAK2 (0.57) TSHRMAPTALDH1A1HSD17B10JAK2
SCHEMBL1833187 0.75 KDM4E (0.48) TSHRMAPTALDH1A1KDM4ENPSR1
SCHEMBL3080180 0.72 L3MBTL1 (0.53) TSHRJAK2JAK3KDM4ERAB9A
SCHEMBL716631 0.72 TSHR (0.50) TSHRMAPTALDH1A1HSD17B10RAB9A
SCHEMBL263628 0.72 TSHR (0.52) TSHRMAPTALDH1A1HSD17B10KDM4E
SCHEMBL11082890 0.71 SMN1; SMN2 (0.63) TSHRMAPTALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099452-A2 TRICARBONYL COMPLEXES WITH TRIDENTATE CHELATORS FOR MYOCARDIUM IMAGING Mallinckrodt Inc. (US) 2009-09-16 EP disclosed
WO-2008061792-A2 TRICARBONYL COMPLEXES WITH TRIDENTATE CHELATORS FOR MYOCARDIUM IMAGING MALLINCKRODT INC. (US) 2008-05-29 WO disclosed
EP-0667868-A1 NEW CEPHEM COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-08-23 EP disclosed
EP-0091130-A2 Cephalosporin derivatives, process for preparing and pharmaceutical compositions containing said compounds DAIICHI SEIYAKU CO., LTD. (JP) 1983-10-12 EP disclosed