SCHEMBL382910

SCHEMBL382910

O=C(Nc1ccccc1)N1CCc2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 1.00
RAB9A P51151 7/20 1.00
SMN1; SMN2 Q16637 6/20 1.00
NFKB1 P19838 4/20 1.00
NFKB2 Q00653 4/20 1.00
RELA Q04206 4/20 1.00
TP53 P04637 4/20 1.00
PKM P14618 3/20 1.00
MAPT P10636 5/20 0.74
MAOB P27338 1/20 0.74
HTR2C P28335 1/20 0.72
HSD17B10 Q99714 1/20 0.66
POLB P06746 1/20 0.64
USP2 O75604 1/20 0.62
NAMPT P43490 1/20 0.61
LMNA P02545 2/20 0.60
ROCK2 O75116 2/20 0.60
ROCK1 Q13464 2/20 0.60
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6350744 0.90 NPC1 (0.81) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL4867471 0.89 TP53 (0.81) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL28367238 0.89 NPC1 (0.79) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL19675330 0.88 NPC1 (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL12692434 0.88 NPC1 (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL28367564 0.88 NPC1 (1.00) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6798342 0.88 NPC1 (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL15879125 0.88 NPC1 (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL4869023 0.88 TP53 (0.78) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL12692444 0.86 RAB9A (1.00) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110878070-B Method for preparing asymmetric urea compound 中国科学院化学研究所 2021-08-31 CN disclosed
CN-110878070-A Method for preparing asymmetric urea compound 中国科学院化学研究所 2020-03-13 CN disclosed
EP-2408744-A1 BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYLGLYCEROL ACYLTRANSFERASE Schering Corporation (US) 2012-01-25 EP disclosed
WO-2010107768-A1 BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYLGLYCEROL ACYLTRANSFERASE SCHERING CORPORATION (US) 2010-09-23 WO disclosed