SCHEMBL3836057

SCHEMBL3836057

CC(C)Oc1cc2c(c(-c3ccc[nH]3)c1)C(=O)NC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.57
KDR P35968 7/20 0.57
TLK2 Q86UE8 2/20 0.42
MAP3K9 P80192 2/20 0.41
MAP3K11 Q16584 2/20 0.41
CDK2 P24941 5/20 0.38
NTRK1 P04629 1/20 0.36
FYN P06241 1/20 0.36
FLT4 P35916 1/20 0.36
MAP3K10 Q02779 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
CDK1 P06493 1/20 0.34
GCK P35557 1/20 0.34
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3840660 0.81 KDR (0.62) AURKAKDRMAP3K9MAP3K11CDK1
SCHEMBL3836059 0.80 AURKA (0.54) AURKAKDRCDK2
SCHEMBL3835796 0.75 MAP3K9 (0.38) AURKAKDRMAP3K9MAP3K11NTRK1
SCHEMBL5328900 0.73 AURKA (1.00) AURKAKDRMAP3K9MAP3K11CDK2
SCHEMBL20992951 0.72 CLK4 (0.47) KDRTLK2MAP3K9MAP3K11NTRK1
SCHEMBL20992953 0.72 MAP3K9 (0.47) TLK2MAP3K9MAP3K11NTRK1FYN
Hydrochloric Acid SCHEMBL3837341 0.71 AURKA (0.56) AURKAKDRCDK2CDK1CA12
SCHEMBL12469307 0.69 AURKA (0.37) AURKAKDRMAP3K9MAP3K11NTRK1
SCHEMBL20992950 0.66 AURKA (0.46) AURKAKDRMAP3K9MAP3K11PIK3CA
SCHEMBL5329803 0.64 KDR (0.77) AURKAKDRCDK1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed