SCHEMBL12469307

SCHEMBL12469307

Cc1nc(-c2cc(OC(C)C)cc3c2C(=O)NC3)[nH]c1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.37
KDR P35968 2/20 0.37
MAP3K9 P80192 2/20 0.36
MAP3K11 Q16584 2/20 0.36
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PIK3R1 P27986 1/20 0.33
NTRK1 P04629 1/20 0.33
FYN P06241 1/20 0.33
FLT4 P35916 1/20 0.33
MAP3K10 Q02779 1/20 0.33
LMNA P02545 1/20 0.32
LRRK2 Q5S007 1/20 0.31
GCK P35557 3/20 0.31
ALDH1A1 P00352 1/20 0.30
MAP3K5 Q99683 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836057 0.69 AURKA (0.57) AURKAKDRMAP3K9MAP3K11PIK3CD
SCHEMBL3840660 0.69 KDR (0.62) AURKAKDRMAP3K9MAP3K11LMNA
SCHEMBL3835796 0.68 MAP3K9 (0.38) AURKAKDRMAP3K9MAP3K11PIK3CD
SCHEMBL12469179 0.66 BRD4 (0.34) AURKAKDR
SCHEMBL20992951 0.65 CLK4 (0.47) KDRMAP3K9MAP3K11PIK3CDPIK3CA
SCHEMBL20992953 0.65 MAP3K9 (0.47) MAP3K9MAP3K11NTRK1FYNFLT4
SCHEMBL15814826 0.59 ALDH1A1 (0.48) PIK3CDPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL743016 0.59 MCL1 (0.59) LMNAALDH1A1
SCHEMBL8466568 0.59 KDR (0.44) AURKAKDRMAP3K9MAP3K11NTRK1
SCHEMBL3839919 0.58 GCK (0.34) MAP3K9MAP3K11NTRK1FYNFLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed