SCHEMBL3836617

SCHEMBL3836617

O=C(O)CC1(NC(=O)OCc2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
HTT P42858 1/20 0.49
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
ALDH1A1 P00352 4/20 0.46
GAA P10253 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1162743 0.93 CTSL (0.45) CTSLCTSBCTSSHTTLMNA
SCHEMBL4110578 0.93 CTSS (0.55) CTSLCTSBCTSSHTTLMNA
SCHEMBL14894910 0.88 NPC1 (0.47) CTSLCTSBCTSSHTTLMNA
SCHEMBL14894968 0.86 CTSL (0.44) CTSLCTSBCTSSHTTLMNA
SCHEMBL381668 0.86 CTSL (0.50) CTSLCTSBCTSSHTTLMNA
SCHEMBL6897899 0.85 HTT (0.54) CTSLCTSBCTSSHTTLMNA
SCHEMBL19442303 0.85 CTSL (0.49) CTSLCTSBCTSSHTTLMNA
SCHEMBL12070062 0.85 CTSL (0.49) CTSLCTSBCTSSHTTLMNA
SCHEMBL16219332 0.85 CTSL (0.52) CTSLCTSBCTSSHTTLMNA
SCHEMBL7950582 0.85 CA12 (0.50) CTSLCTSBCTSSHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149213-A2 NOVEL DERIVATIVE HAVING INHIBITORY ACTIVITY AGAINST 11Β-HSD1, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT 주식회사 이큐스앤자루 (KR) 2011-12-01 WO disclosed
EP-1658267-B1 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2009-10-14 EP disclosed
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed