SCHEMBL3837047

SCHEMBL3837047

CCc1cccc(CC)c1-c1nc(C)c(CN2CCOc3ccc(C)nc32)c(N2CCN(C(=O)O)CC2)n1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 1/20 0.33
GBA1 P04062 1/20 0.31
MAPK1 P28482 1/20 0.30
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NUDT1 P36639 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3509664 0.94 PTGER3 (0.32) PTGER3GBA1
SCHEMBL62739 0.89 GBA1 (0.37) GBA1
SCHEMBL62176 0.89 PTGER3 (0.31) PTGER3ALDH1A1MAPTNUDT1
SCHEMBL63143 0.88 PIK3CD (0.35) PTGER3MEN1KMT2AALDH1A1NUDT1
SCHEMBL62172 0.87 MEN1 (0.34) MAPK1MEN1KMT2A
SCHEMBL62683 0.87 TSHR (0.36) PTGER3MAPK1MEN1KMT2AALDH1A1
SCHEMBL62209 0.86 GBA1 (0.31) GBA1NUDT1
SCHEMBL61175 0.85 CYP11B2 (0.41) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL61696 0.85 PIK3CD (0.33) PTGER3
SCHEMBL61296 0.77 ELANE (0.33) MAPK1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745033-A4 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORP (US) 2009-08-26 EP claimed
EP-1745033-A2 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORPORATION (US) 2007-01-24 EP claimed
WO-2005110416-A2 4,5-DISUBSTITUTED-2-ARYL PYRIMIDINES NEUROGEN CORPORATION (US) 2005-11-24 WO claimed