SCHEMBL61696

SCHEMBL61696

CCc1cccc(CC)c1-c1nc(C)c(CN2CCOc3ccc(C)nc32)c(N2CCN(C(=O)C(=O)O)C(C)C2)n1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 3/20 0.33
SMO Q99835 3/20 0.31
KDM4E B2RXH2 1/20 0.31
CXCR3 P49682 1/20 0.31
LIMK2 P53671 1/20 0.31
SCD5 Q86SK9 1/20 0.31
PIK3R1 P27986 1/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30
CHRM1 P11229 1/20 0.30
HTR1A P08908 2/20 0.30
HTR1D P28221 2/20 0.30
HTR1B P28222 2/20 0.30
SLC6A4 P31645 2/20 0.30
KCNH2 Q12809 2/20 0.30
PTGER3 P43115 1/20 0.30
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3509664 0.89 PTGER3 (0.32) PTGER3
SCHEMBL3837047 0.85 PTGER3 (0.33) PTGER3
SCHEMBL62176 0.82 PTGER3 (0.31) PTGER3
SCHEMBL62683 0.82 TSHR (0.36) KDM4EPTGER3
SCHEMBL61695 0.81 PTGER3 (0.32) PTGER3
SCHEMBL63143 0.81 PIK3CD (0.35) PIK3CDKDM4EHTR1AHTR1DHTR1B
SCHEMBL61440 0.81 OGA (0.33) PIK3CD
SCHEMBL62172 0.81 MEN1 (0.34) KDM4EHTR1ASLC6A4KCNH2
SCHEMBL62209 0.80 GBA1 (0.31) KDM4E
SCHEMBL63402 0.80 ADRA2A (0.34) KDM4EHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129395-B2 4,5-disubstituted-2-aryl pyrimidines NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-03-06 US disclosed