SCHEMBL383876

SCHEMBL383876

c1cnc2nc(NC3CCNCC3)[nH]c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.50
KCNH2 Q12809 1/20 0.45
NUDT1 P36639 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
PIM1 P11309 2/20 0.43
AURKA O14965 2/20 0.41
RIPK1 Q13546 1/20 0.40
METAP2 P50579 1/20 0.40
METAP1 P53582 1/20 0.40
PDE5A O76074 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
ALOX15 P16050 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9690509 0.94 PIM1 (0.46) PTPN11KCNH2NUDT1HRH3PIM1
SCHEMBL9044459 0.78 PTPN11 (0.48) PTPN11HRH3PIM1USP2ALDH1A1
SCHEMBL382481 0.78 JAK1 (0.54) KCNH2RIPK1
Bromide SCHEMBL3874715 0.77 JAK1 (0.53) KCNH2RIPK1
Hydrochloric Acid SCHEMBL5007369 0.77 JAK1 (0.53) KCNH2RIPK1
Hydrochloric Acid SCHEMBL8130344 0.77 JAK1 (0.53) KCNH2RIPK1
SCHEMBL14447540 0.75 NPY5R (0.53) NUDT1AURKAMETAP2METAP1PDE5A
SCHEMBL9535416 0.74 PIM1 (0.48) PTPN11HRH3PIM1RIPK1USP2
SCHEMBL417542 0.73 NOS2 (0.61) ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL9689129 0.73 PIM1 (0.47) PTPN11HRH3PIM1RIPK1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US disclosed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP disclosed