SCHEMBL3840778

SCHEMBL3840778

Cc1ccc(-c2ccc(OC3CN4CCC3CC4)nn2)c(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.53
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALDH1A1 P00352 1/20 0.37
LSS P48449 1/20 0.37
GLA P06280 1/20 0.36
TSHR P16473 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
GAA P10253 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3840773 1.00 CHRNA7 (0.53) CHRNA7CYP1A2CYP2D6ALDH1A1LSS
SCHEMBL1459282 0.87 CHRNA7 (0.53) CHRNA7CYP1A2CYP2D6ALDH1A1
SCHEMBL1459280 0.87 CHRNA7 (0.53) CHRNA7CYP1A2CYP2D6ALDH1A1
SCHEMBL3839223 0.84 CHRNA7 (0.53) CHRNA7CYP1A2CYP2D6ALDH1A1
SCHEMBL3839228 0.84 CHRNA7 (0.53) CHRNA7CYP1A2CYP2D6ALDH1A1
SCHEMBL3840517 0.84 CHRNA7 (0.54) CHRNA7LSSGLAGAAATM
SCHEMBL3840519 0.84 CHRNA7 (0.54) CHRNA7LSSGLAGAAATM
SCHEMBL3842064 0.81 CHRNA7 (0.47) CHRNA7CYP1A2CYP2D6
SCHEMBL3839401 0.81 CHRNA7 (0.47) CHRNA7CYP1A2CYP2D6
SCHEMBL3839400 0.81 CHRNA7 (0.69) CHRNA7CYP1A2CYP2D6LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8236803-B2 Aza-bicycloalkyl ethers and their use as alpha7-nAChR agonists NOVARTIS AG (CH) 2012-08-07 US claimed
EP-1537104-B1 AZA-BICYCLOALKYL ETHERS AND THEIR USE AS ALPHA7-NACHR AGONISTS NOVARTIS AG (CH) 2009-11-11 EP claimed
EP-1537104-B1 AZA-BICYCLOALKYL ETHERS AND THEIR USE AS ALPHA7-NACHR AGONISTS NOVARTIS AG (CH) 2009-11-11 EP disclosed