SCHEMBL3841879

SCHEMBL3841879

CN(C)c1ccc(O)c(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
MAPK1 P28482 2/20 0.48
EP300 Q09472 1/20 0.47
KAT2B Q92831 1/20 0.47
KAT8 Q9H7Z6 1/20 0.47
GAA P10253 3/20 0.38
KMT2A Q03164 2/20 0.38
APP P05067 7/20 0.37
ESR1 P03372 1/20 0.36
TSHR P16473 4/20 0.36
FABP4 P15090 1/20 0.33
HSD17B10 Q99714 3/20 0.32
HPGD P15428 2/20 0.32
HSP90AA1 P07900 1/20 0.32
LMNA P02545 2/20 0.32
CYP1A2 P05177 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPT P10636 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2443752 0.84 GAA (0.46) CYP3A4MAPK1EP300KAT2BKAT8
SCHEMBL15934243 0.79 TSHR (0.50) CYP3A4MAPK1EP300KAT2BKAT8
SCHEMBL28153042 0.76 HPGD (0.48) CYP3A4MAPK1EP300KAT2BKAT8
SCHEMBL68064 0.76 CYP3A4 (0.75) CYP3A4MAPK1KMT2AESR1TSHR
SCHEMBL31392414 0.76 CYP3A4 (0.75) CYP3A4MAPK1KMT2AESR1TSHR
SCHEMBL7743436 0.76 CYP3A4 (0.75) CYP3A4MAPK1KMT2AESR1TSHR
SCHEMBL8927868 0.75 CYP3A4 (0.40) CYP3A4MAPK1EP300KAT2BKAT8
SCHEMBL3222106 0.70 HSD17B10 (0.50) CYP3A4MAPK1EP300KAT2BKAT8
SCHEMBL3786708 0.69 GAA (0.52) CYP3A4MAPK1GAAKMT2ATSHR
SCHEMBL11036013 0.69 CYP3A4 (0.57) CYP3A4MAPK1GAAESR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088861-A2 BENZIMIDAZOLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-08-19 EP disclosed
WO-2008051533-A2 BENZIMIDAZOLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed