SCHEMBL3843503

SCHEMBL3843503

Fc1ccc(C(F)(F)F)cc1-c1ccc(O[C@H]2CN3CCC2CC3)nn1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.51
KDM1A O60341 1/20 0.39
IL1B P01584 1/20 0.38
NLRP3 Q96P20 1/20 0.38
MPL P40238 1/20 0.36
HTR3A P46098 1/20 0.36
CHRM2 P08172 2/20 0.34
CHRM1 P11229 2/20 0.34
CHRM3 P20309 2/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3843507 1.00 CHRNA7 (0.51) CHRNA7KDM1AIL1BNLRP3MPL
SCHEMBL3840240 0.87 CHRNA7 (0.54) CHRNA7CHRM2CHRM1CHRM3CHRM4
SCHEMBL3840243 0.87 CHRNA7 (0.54) CHRNA7CHRM2CHRM1CHRM3CHRM4
SCHEMBL3839223 0.85 CHRNA7 (0.53) CHRNA7CHRM2CHRM1CHRM3
SCHEMBL3839228 0.85 CHRNA7 (0.53) CHRNA7CHRM2CHRM1CHRM3
SCHEMBL3840352 0.83 CHRNA7 (0.61) CHRNA7IL1BNLRP3CHRM2CHRM1
SCHEMBL3840349 0.83 CHRNA7 (0.61) CHRNA7IL1BNLRP3CHRM2CHRM1
SCHEMBL3844594 0.82 CHRNA7 (0.54) CHRNA7KDM1AMPL
SCHEMBL3840541 0.82 CHRNA7 (0.54) CHRNA7CHRM2CHRM1CHRM3CHRM4
SCHEMBL3840537 0.82 CHRNA7 (0.54) CHRNA7CHRM2CHRM1CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8236803-B2 Aza-bicycloalkyl ethers and their use as alpha7-nAChR agonists NOVARTIS AG (CH) 2012-08-07 US claimed
EP-1537104-B1 AZA-BICYCLOALKYL ETHERS AND THEIR USE AS ALPHA7-NACHR AGONISTS NOVARTIS AG (CH) 2009-11-11 EP claimed