SCHEMBL3845506

SCHEMBL3845506

CCCCCCCn1nc(NCCCc2ccc(SC(C)(CCC)C(=O)O)cc2)c(=O)n(C)c1=O

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.37
S1PR3 Q99500 4/20 0.37
S1PR2 O95136 3/20 0.37
S1PR4 O95977 2/20 0.37
PPARG P37231 6/20 0.34
PPARA Q07869 6/20 0.34
PPARD Q03181 5/20 0.34
TRPA1 O75762 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
SMPD1 P17405 1/20 0.32
CNR1 P21554 2/20 0.31
CNR2 P34972 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3851231 0.96 S1PR1 (0.35) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3844823 0.91 PPARG (0.42) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3840985 0.88 PPARG (0.36) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3285318 0.86 PPARG (0.41) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3288469 0.84 TLR7 (0.34) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3845660 0.83 S1PR1 (0.36) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3849410 0.81 PPARG (0.40) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3840711 0.80 MAOA (0.33) S1PR1S1PR3S1PR2S1PR4PPARG
SCHEMBL3284220 0.80 MAPT (0.34) PPARGPPARAPPARDTRPA1MAOA
SCHEMBL3841112 0.80 PPARG (0.39) PPARGPPARAPPARDSMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856065-B1 1,2,4-TRIAZINE DERIVATIVES, PREPARATION AND USE THEREOF IN HUMAN THERAPY PF MEDICAMENT (FR) 2009-11-11 EP claimed