SCHEMBL3846729

SCHEMBL3846729

O=C(Nc1ccc(Cl)cn1)c1ccc(-c2cnc3ccc(-c4cn[nH]c4)cn23)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
FLT3 P36888 2/20 0.41
NRAS P01111 1/20 0.41
SORT1 Q99523 1/20 0.41
F10 P00742 3/20 0.41
KCNH2 Q12809 2/20 0.41
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
BRD4 O60885 1/20 0.39
CSNK1D P48730 1/20 0.39
CSNK1E P49674 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
KIT P10721 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3847294 0.99 SMN1; SMN2 (0.45) SMN1; SMN2TDP1FLT3NRASSORT1
Hydrochloric Acid SCHEMBL3849166 0.90 FLT3 (0.42) FLT3NRASKITROCK2ROCK1
SCHEMBL3856718 0.90 NPC1 (0.46) SMN1; SMN2FLT3NRASSORT1NPC1
Hydrochloric Acid SCHEMBL5852371 0.89 NPC1 (0.45) SMN1; SMN2FLT3NRASSORT1NPC1
SCHEMBL4713522 0.87 CHEK1 (0.42) FLT3NRASCSNK1DCSNK1EKIT
SCHEMBL4711686 0.87 FLT3 (0.40) FLT3NRASKITROCK2ROCK1
Hydrochloric Acid SCHEMBL3846953 0.87 KIT (0.39) SMN1; SMN2FLT3NRASNPC1RAB9A
Hydrochloric Acid SCHEMBL3855591 0.87 CHEK1 (0.41) FLT3NRASCSNK1DCSNK1EKIT
Hydrochloric Acid SCHEMBL3846948 0.87 FLT3 (0.39) FLT3NRASKITROCK2ROCK1
Hydrochloric Acid SCHEMBL3850563 0.85 FLT3 (0.41) FLT3NRASNPC1RAB9AKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP claimed
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed