SCHEMBL3856718

SCHEMBL3856718

Cc1ccc(NC(=O)c2ccc(-c3cnc4ccc(-c5cn[nH]c5)cn34)cc2F)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
TP53 P04637 2/20 0.46
GAA P10253 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CLK1 P49759 2/20 0.43
CLK2 P49760 2/20 0.43
FLT3 P36888 2/20 0.41
NRAS P01111 1/20 0.41
MAP3K5 Q99683 1/20 0.41
SORT1 Q99523 1/20 0.41
KIT P10721 1/20 0.41
MITF O75030 1/20 0.41
PTK6 Q13882 1/20 0.40
AURKB Q96GD4 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5852371 0.99 NPC1 (0.45) NPC1RAB9ATP53GAAKDM4E
Hydrochloric Acid SCHEMBL3849166 0.90 FLT3 (0.42) CLK1CLK2FLT3NRASMAP3K5
SCHEMBL3846729 0.90 SMN1; SMN2 (0.46) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL4713522 0.89 CHEK1 (0.42) CLK1CLK2FLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL3847294 0.89 SMN1; SMN2 (0.45) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL4715804 0.89 LOXL2 (0.43) NPC1RAB9ASMN1; SMN2CLK1CLK2
Hydrochloric Acid SCHEMBL3855591 0.88 CHEK1 (0.41) CLK1CLK2FLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL3847724 0.88 LOXL2 (0.42) NPC1RAB9ASMN1; SMN2CLK1CLK2
SCHEMBL4711686 0.87 FLT3 (0.40) CLK1CLK2FLT3NRASMAP3K5
Hydrochloric Acid SCHEMBL3846948 0.87 FLT3 (0.39) CLK1CLK2FLT3NRASMAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed