SCHEMBL4711686

SCHEMBL4711686

C=Cc1ccc(NC(=O)c2ccc(-c3cnc4ccc(-c5cn[nH]c5)cn34)cc2F)nc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.40
NRAS P01111 1/20 0.40
CHEK1 O14757 4/20 0.38
CHEK2 O96017 3/20 0.38
ABL1 P00519 2/20 0.38
MAPK1 P28482 1/20 0.37
IKBKB O14920 5/20 0.37
KIT P10721 1/20 0.37
ROCK2 O75116 2/20 0.37
ROCK1 Q13464 2/20 0.37
MELK Q14680 1/20 0.36
MAP3K5 Q99683 1/20 0.36
CLK1 P49759 2/20 0.36
CLK2 P49760 2/20 0.36
PTK6 Q13882 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3846948 0.99 FLT3 (0.39) FLT3NRASCHEK1CHEK2ABL1
Hydrochloric Acid SCHEMBL3849166 0.88 FLT3 (0.42) FLT3NRASCHEK1CHEK2ABL1
SCHEMBL3856718 0.87 NPC1 (0.46) FLT3NRASKITROCK2ROCK1
SCHEMBL3846729 0.87 SMN1; SMN2 (0.46) FLT3NRASCHEK1CHEK2ABL1
SCHEMBL4713522 0.87 CHEK1 (0.42) FLT3NRASCHEK1CHEK2ABL1
Hydrochloric Acid SCHEMBL3847294 0.87 SMN1; SMN2 (0.45) FLT3NRASCHEK1CHEK2ABL1
Hydrochloric Acid SCHEMBL5852371 0.87 NPC1 (0.45) FLT3NRASKITROCK2ROCK1
Hydrochloric Acid SCHEMBL3855591 0.86 CHEK1 (0.41) FLT3NRASCHEK1CHEK2ABL1
SCHEMBL4715804 0.82 LOXL2 (0.43) FLT3NRASCHEK1CHEK2ABL1
SCHEMBL3846503 0.81 CLK1 (0.37) MAPK1IKBKBCLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP claimed