SCHEMBL3847251

SCHEMBL3847251

C=C[C@]12CC[C@]3(C)[C@@H](F)[C@H](O[Si](C)(C)C(C)(C)C)C[C@H]3[C@@H]1CCc1cc(O[Si](C)(C)C(C)(C)C)ccc12

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3844568 0.90 LMNA (0.31)
SCHEMBL5156005 0.86 ESR1 (0.32)
SCHEMBL3846173 0.83 ESR2 (0.43)
SCHEMBL3848340 0.82 STS (0.31)
SCHEMBL3847345 0.81 RORC (0.33)
SCHEMBL3854474 0.79 ESR1 (0.32)
SCHEMBL3854471 0.79 ESR1 (0.32)
SCHEMBL3848400 0.79 STS (0.31)
SCHEMBL6028199 0.70 ESR1 (0.44)
SCHEMBL6027234 0.70 ESR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2039702-A2 Prodrugs erbeta-selective substances, method for their production and pharmaceutical compounds containing these compositions Bayer Schering Pharma Aktiengesellschaft (DE) 2009-03-25 EP disclosed
US-20070123500-A1 Prodrugs of ERbeta-selective substances, processes for their preparation and pharmaceutical compositions comprising these compounds BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-05-31 US disclosed