SCHEMBL3847323

SCHEMBL3847323

COc1ccc2nc(OCc3ccccc3)nc(Nc3ccc(Br)cc3F)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.49
ERBB2 P04626 1/20 0.49
CLK1 P49759 1/20 0.47
KDR P35968 4/20 0.47
RET P07949 1/20 0.47
KIF5B P33176 1/20 0.47
NPC1 O15118 1/20 0.44
NCOA1 Q15788 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
MAPT P10636 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
POLB P06746 3/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PDE5A O76074 2/20 0.40
TBXAS1 P24557 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138839 0.81 EGFR (0.43) EGFRERBB2NPC1MAPTKMT2A
Hydrochloric Acid SCHEMBL1893474 0.78 KDR (0.42) EGFRCLK1KDRRETKIF5B
SCHEMBL29368280 0.77 EGFR (0.72) EGFRCLK1KDRRETKIF5B
SCHEMBL159652 0.75 KDR (0.80) EGFRERBB2KDRRETKIF5B
Hydrochloric Acid SCHEMBL1468204 0.74 KDR (0.78) EGFRERBB2KDRRETKIF5B
SCHEMBL7499766 0.74 ALDH1A1 (0.51) EGFRERBB2NPC1MAPTKMT2A
Hydrochloric Acid SCHEMBL8708549 0.73 KDR (0.49) EGFRERBB2KDRRETKIF5B
SCHEMBL6471210 0.73 EGFR (0.50) EGFRERBB2NPC1MAPTKMT2A
SCHEMBL31006585 0.72 NPC1 (0.76) EGFRCLK1KDRRETKIF5B
SCHEMBL29283856 0.72 NPC1 (0.76) EGFRCLK1KDRRETKIF5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943240-B1 CHEMICAL PROCESS ASTRAZENECA AB (SE) 2009-11-11 EP disclosed