SCHEMBL3848867

SCHEMBL3848867

CSc1cc(C2CCN(c3ccnc4ccc(Br)cc34)CC2)c(C=O)s1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 3/20 0.47
CHRM4 P08173 1/20 0.35
SLC22A12 Q96S37 6/20 0.34
HTT P42858 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
IDE P14735 1/20 0.31
TGFBR1 P36897 1/20 0.30
NMT1 P30419 2/20 0.30
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30
HTR7 P34969 1/20 0.30
HTR6 P50406 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3851360 0.85 HTT (0.49) CHRM4HTTALDH1A1NPSR1MEN1
SCHEMBL3848117 0.82 NCF1 (0.49) NCF1CHRM4SLC22A12HTTALDH1A1
SCHEMBL3848807 0.81 NCF1 (0.48) NCF1CHRM4SLC22A12HTTTGFBR1
SCHEMBL3856295 0.77 NCF1 (0.47) NCF1CHRM4SLC22A12HTTTGFBR1
SCHEMBL3846163 0.77 NCF1 (0.52) NCF1CHRM4HTR1A
SCHEMBL3848381 0.75 NCF1 (0.47) NCF1CHRM4SLC22A12ALDH1A1IDE
SCHEMBL21190487 0.70 NCF1 (0.67) NCF1CHRM4SLC22A12HTTALDH1A1
SCHEMBL1544187 0.70 NCF1 (0.62) NCF1CHRM4SLC22A12HTTALDH1A1
SCHEMBL3848120 0.69 NCF1 (0.50) NCF1CHRM4SLC22A12ALDH1A1MEN1
SCHEMBL3845241 0.69 NCF1 (0.61) NCF1CHRM4SLC22A12ALDH1A1IDE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed