SCHEMBL3845241

SCHEMBL3845241

O=C(O)C1CCN(c2ccnc3ccc(Br)cc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.61
PPARG P37231 1/20 0.57
ATM Q13315 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57
NCOR2 Q9Y618 1/20 0.57
KDM4E B2RXH2 2/20 0.46
CYP2C19 P33261 1/20 0.46
SLC22A12 Q96S37 4/20 0.45
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
IDE P14735 1/20 0.42
NEK2 P51955 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 2/20 0.41
CYP2C9 P11712 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14145384 0.89 NCF1 (0.60) NCF1PPARGATMRXFP1NCOR2
SCHEMBL3848428 0.86 NCF1 (0.56) NCF1PPARGATMRXFP1NCOR2
SCHEMBL3846166 0.83 NCF1 (0.53) NCF1KDM4EALDH1A1POLBGAA
SCHEMBL3846599 0.83 ALDH1A1 (0.56) NCF1KDM4EALDH1A1IDEMAPK1
SCHEMBL1777402 0.82 NCF1 (0.64) NCF1SLC22A12ALDH1A1IDEMAPK1
SCHEMBL21190487 0.82 NCF1 (0.67) NCF1SLC22A12ALDH1A1KMT2AHSD17B10
SCHEMBL19000116 0.82 ADRB2 (0.57) NCF1KDM4ECYP2C19ALDH1A1IDE
SCHEMBL3848120 0.81 NCF1 (0.50) NCF1PPARGATMRXFP1NCOR2
SCHEMBL14145469 0.81 LMNA (0.53) NCF1RXFP1ALDH1A1KMT2ACHRM4
SCHEMBL3848733 0.81 NCF1 (0.50) NCF1ATMALDH1A1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed