SCHEMBL3849461

SCHEMBL3849461

CN(c1ccnn1-c1ccccc1)S(=O)(=O)c1ccc(N)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C18 P33260 16/20 1.00
CYP2C9 P11712 16/20 1.00
CYP2C8 P10632 13/20 1.00
CYP2C19 P33261 13/20 0.79
LMNA P02545 1/20 0.57
POLB P06746 1/20 0.57
CYP3A4 P08684 1/20 0.57
TSHR P16473 1/20 0.57
NFKB1 P19838 1/20 0.57
THPO P40225 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
HSD17B10 Q99714 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
C1R P00736 1/20 0.47
PRSS1 P07477 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL896130 0.88 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C8CYP2C19C1R
SCHEMBL3845016 0.84 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C8CYP2C19LMNA
SCHEMBL3847126 0.82 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C8CYP2C19LMNA
Sulfaphenazole SCHEMBL122040 0.73 CYP2C9 (1.00) CYP2C18CYP2C9CYP2C8CYP2C19LMNA
SCHEMBL2518894 0.72 CA12 (0.71) CYP2C18CYP2C9CYP2C8LMNATSHR
SCHEMBL1004589 0.70 CYP2C9 (0.54) CYP2C18CYP2C9CYP2C8CYP2C19LMNA
Sulfaphenazole SCHEMBL28086445 0.68 CYP2C9 (0.80) CYP2C18CYP2C9CYP2C8CYP2C19LMNA
SCHEMBL5121853 0.66 C5AR1 (0.59) CYP2C18CYP2C9CYP2C8LMNACYP3A4
SCHEMBL5121845 0.66 MAPT (0.68) CYP2C18CYP2C9CYP2C8LMNACYP3A4
SCHEMBL2841054 0.66 CYP2C18 (0.50) CYP2C18CYP2C9CYP2C8CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2011489-A2 Method to inhibit ischemia and reperfusion injury Gottlieb, Roberta (US) 2009-01-07 EP disclosed
EP-1523310-A2 METHOD TO INHIBIT ISCHEMIA AND REPERFUSION INJURY The Scripps Research Institute (US) 2005-04-20 EP disclosed
WO-2004004702-A2 METHOD TO INHIBIT ISCHEMIA AND REPERFUSION INJURY THE SCRIPPS RESEARCH INSTITUTE (US) 2004-01-15 WO disclosed