SCHEMBL896130

SCHEMBL896130

Cc1ccc(S(=O)(=O)N(C)c2ccnn2-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C18 P33260 13/20 1.00
CYP2C9 P11712 12/20 1.00
CYP2C19 P33261 10/20 1.00
CYP2C8 P10632 12/20 0.79
CA12 O43570 1/20 0.54
CA9 Q16790 1/20 0.54
C5AR1 P21730 1/20 0.51
MAPT P10636 1/20 0.46
MCOLN3 Q8TDD5 1/20 0.46
C1R P00736 1/20 0.46
PRSS1 P07477 1/20 0.46
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3849461 0.88 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C19CYP2C8C1R
SCHEMBL3845016 0.72 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C19CYP2C8
SCHEMBL3822617 0.71 CA12 (1.00) CA12CA9C5AR1MAPTMCOLN3
SCHEMBL3847126 0.70 CYP2C18 (1.00) CYP2C18CYP2C9CYP2C19CYP2C8
SCHEMBL8553556 0.69 CYP2C9 (0.70) CYP2C18CYP2C9CYP2C19CYP2C8ALDH1A1
SCHEMBL11910521 0.68 CA12 (0.86) CA12CA9C5AR1MAPTMCOLN3
SCHEMBL2841054 0.67 CYP2C18 (0.50) CYP2C18CYP2C9CYP2C19CYP2C8CA12
SCHEMBL15834271 0.66 CYP2C9 (0.69) CYP2C18CYP2C9CYP2C19CYP2C8ALDH1A1
SCHEMBL14973952 0.65 CYP2C18 (0.48) CYP2C18CYP2C9CYP2C19CYP2C8
SCHEMBL7150548 0.65 C5AR1 (0.83) CYP2C18CYP2C9CYP2C19CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8793078-B2 Method for predicting activation energy using atomic fingerprint descriptor or atomic descriptor BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2014-07-29 US disclosed
US-20120084012-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING ATOMIC FINGERPRINT DESCRIPTOR OR ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2012-04-05 US disclosed
US-20110213558-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2011-09-01 US disclosed
EP-2354987-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR Bioinformatics&Molecular Design Research Center (KR) 2011-08-10 EP disclosed
WO-2010056053-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR 사단법인 분자설계연구소 (KR) 2010-05-20 WO disclosed