SCHEMBL3852629

SCHEMBL3852629

CN(C)S(=O)(=O)N1CCN(c2ccnc3ccc(Br)cc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.58
SORD Q00796 4/20 0.47
ALDH1A1 P00352 7/20 0.46
MCOLN3 Q8TDD5 1/20 0.46
SLC22A12 Q96S37 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 4/20 0.43
HTT P42858 4/20 0.43
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3847734 0.79 NCF1 (0.70) NCF1ALDH1A1SLC22A12NPSR1HTT
SCHEMBL3846343 0.79 NCF1 (0.58) NCF1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL22715673 0.78 NCF1 (0.76) NCF1ALDH1A1SLC22A12NPSR1HTT
SCHEMBL29472100 0.78 NCF1 (0.76) NCF1ALDH1A1SLC22A12NPSR1HTT
SCHEMBL3850039 0.77 SORD (0.40) NCF1SORDALDH1A1MCOLN3NPSR1
SCHEMBL731691 0.76 NCF1 (0.74) NCF1ALDH1A1SLC22A12NPSR1HTT
SCHEMBL1777402 0.75 NCF1 (0.64) NCF1ALDH1A1SLC22A12SMN1; SMN2MEN1
SCHEMBL30734145 0.75 NCF1 (0.67) NCF1ALDH1A1NPSR1KDM4EHTT
SCHEMBL3848428 0.74 NCF1 (0.56) NCF1ALDH1A1SLC22A12
SCHEMBL3847838 0.74 SORD (0.38) NCF1SORDALDH1A1MCOLN3NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed