SCHEMBL3853772

SCHEMBL3853772

CN(CCc1c[nH]c2ccccc12)Cc1cc2c(c(-c3cc4cc(CN5CCCCC5)ccc4[nH]3)c1)C(=O)NC2

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.42
KDR P35968 2/20 0.42
CHEK1 O14757 12/20 0.41
HRH3 Q9Y5N1 3/20 0.41
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3887524 0.83 KDR (0.49) AURKAKDRCHEK1
Hydrochloric Acid SCHEMBL3874594 0.82 CHEK1 (0.49) AURKAKDRCHEK1
SCHEMBL3859270 0.81 AURKA (0.44) AURKAKDRCHEK1
SCHEMBL3839644 0.81 HRH3 (0.37) HRH3BCHEACHELMNAHTT
SCHEMBL3839118 0.80 CHEK1 (0.49) AURKAKDRCHEK1
SCHEMBL3837181 0.76 CHEK1 (0.56) AURKAKDRCHEK1
Hydrochloric Acid SCHEMBL3856617 0.75 AURKA (0.51) AURKAKDRCHEK1
SCHEMBL3839156 0.75 CHEK1 (0.56) AURKAKDRCHEK1
SCHEMBL3839022 0.75 CHEK1 (0.63) AURKAKDRCHEK1
Hydrochloric Acid SCHEMBL3841238 0.74 CHEK1 (0.49) AURKAKDRCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed