SCHEMBL3887524

SCHEMBL3887524

COCCN(C)Cc1cc2c(c(-c3cc4cc(CN5CCCCC5)ccc4[nH]3)c1)C(=O)NC2

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.49
AURKA O14965 6/20 0.49
CHEK1 O14757 13/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3874594 0.87 CHEK1 (0.49) KDRAURKACHEK1
SCHEMBL3839118 0.86 CHEK1 (0.49) KDRAURKACHEK1
SCHEMBL3887530 0.84 AURKA (0.49) KDRAURKACHEK1
SCHEMBL3859270 0.83 AURKA (0.44) KDRAURKACHEK1
SCHEMBL3853772 0.83 AURKA (0.42) KDRAURKACHEK1
SCHEMBL3837181 0.81 CHEK1 (0.56) KDRAURKACHEK1
SCHEMBL3839022 0.80 CHEK1 (0.63) KDRAURKACHEK1
SCHEMBL3839156 0.80 CHEK1 (0.56) KDRAURKACHEK1
Hydrochloric Acid SCHEMBL3841238 0.79 CHEK1 (0.49) KDRAURKACHEK1
Hydrochloric Acid SCHEMBL3854182 0.79 AURKA (0.46) KDRAURKACHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed