SCHEMBL3856445

SCHEMBL3856445

N#Cc1cc(Cl)ccc1OC(N)=O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.45
MRGPRX4 Q96LA9 1/20 0.45
KDM4E B2RXH2 2/20 0.43
VCAM1 P19320 1/20 0.42
CYP2D6 P10635 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SYK P43405 1/20 0.41
ADRA1D P25100 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
XDH P47989 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
ALDH1A1 P00352 2/20 0.38
USP2 O75604 1/20 0.38
HPGD P15428 1/20 0.38
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28738819 0.90 NOS2 (0.48) NOS2MRGPRX4KDM4EVCAM1CYP2D6
SCHEMBL6175873 0.83 MAOB (0.47) NOS2MRGPRX4KDM4EVCAM1MAOA
SCHEMBL27336403 0.81 PTGDR2 (0.40) MRGPRX4KDM4EPTGDR2ALDH1A1USP2
SCHEMBL28738821 0.80 AAK1 (0.42) KDM4EMAOAMAOBXDHPTGDR2
SCHEMBL28305946 0.80 FFAR1 (0.43) KDM4EMAOAMAOBXDHALDH1A1
SCHEMBL1853203 0.80 PTGDR2 (0.51) NOS2MRGPRX4PTGDR2MAPT
SCHEMBL8799276 0.79 NOS2 (0.43) NOS2MRGPRX4KDM4EVCAM1CYP2D6
SCHEMBL29728508 0.78 KMT2A (0.42) KDM4EALDH1A1HPGDMEN1MAPT
SCHEMBL8861735 0.77 KMT2A (0.57) MRGPRX4SLC6A2SLC6A4ALDH1A1HPGD
SCHEMBL31441456 0.75 MAOA (0.61) NOS2MRGPRX4KDM4EVCAM1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380718-B Acylation method of aniline compound 河南农业大学 2022-09-30 CN disclosed
CN-114380718-A Acylation method of aniline compound 河南农业大学 2022-04-22 CN disclosed
US-8481569-B2 Iminopyridine derivatives and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-07-09 US disclosed
WO-2009131245-A1 IMINOPYRIDINE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-29 WO disclosed