SCHEMBL3856818

SCHEMBL3856818

CC1CC(C#N)(c2cc(F)ccc2-c2ccc(Br)cc2)C(Cc2ccccc2)CN1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.33
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073736 0.88 PTGS2 (0.38)
SCHEMBL3853509 0.88 PTGS2 (0.38)
SCHEMBL2817918 0.72 SIGMAR1 (0.43)
SCHEMBL2817921 0.72 SIGMAR1 (0.43)
SCHEMBL10073907 0.59 CTSC (0.43) CTSCMAPT
SCHEMBL1773966 0.54 TTR (0.46)
SCHEMBL31649854 0.53 KDM1A (0.32)
SCHEMBL31650647 0.53 KDM1A (0.32)
Benzyl Alcohol SCHEMBL28201559 0.53 TSHR (0.58) NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL26987794 0.53 KDM1A (0.37) NPC1POLBRAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117309-A1 BICYCLIC SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE Merck & Co., Inc. (US) 2009-11-18 EP disclosed
WO-2008085509-A1 BICYCLIC SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2008-07-17 WO disclosed