SCHEMBL3864255

SCHEMBL3864255

O=C(O)CCNNS(=O)(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
TBXA2R P21731 2/20 0.57
BCAT1 P54687 1/20 0.51
KAT6A Q92794 1/20 0.50
MAPT P10636 1/20 0.49
ATM Q13315 1/20 0.49
GAA P10253 2/20 0.47
MMP9 P14780 2/20 0.47
MMP8 P22894 2/20 0.47
MMP13 P45452 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459653 0.85 ALDH1A1 (0.56) ALDH1A1MAPTGAAMMP9MMP8
SCHEMBL1200801 0.81 ALDH1A1 (0.75) ALDH1A1TBXA2RMAPTATMGAA
SCHEMBL28339828 0.81 BCAT1 (0.55) ALDH1A1TBXA2RBCAT1KAT6AMAPT
SCHEMBL7980857 0.79 BCAT1 (0.45) ALDH1A1TBXA2RBCAT1KAT6AMAPT
Hydrazine SCHEMBL11854301 0.79 ALDH1A1 (0.71) ALDH1A1TBXA2RMAPTATMGAA
SCHEMBL28150870 0.78 SMN1; SMN2 (0.50) ALDH1A1BCAT1KAT6AGAAMMP9
Hydrochloric Acid SCHEMBL7447734 0.78 BCAT1 (0.44) ALDH1A1TBXA2RBCAT1KAT6AMAPT
SCHEMBL15482049 0.77 CYP2C19 (0.59) ALDH1A1TBXA2RBCAT1KAT6AGAA
SCHEMBL911198 0.75 ALDH1A1 (0.87) ALDH1A1TBXA2RMAPTATMGAA
SCHEMBL11829145 0.75 BCAT1 (0.61) ALDH1A1BCAT1KAT6AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1044001-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2003-01-29 EP disclosed
EP-1007026-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2002-08-07 EP disclosed
EP-1100506-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2002-06-26 EP disclosed
EP-1105389-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2001-10-17 EP disclosed
EP-1105389-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2001-06-13 EP disclosed
EP-1100506-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2001-05-23 EP disclosed
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
EP-1044001-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-18 EP disclosed
WO-2000009503-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-02-24 WO disclosed
WO-2000006169-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-02-10 WO disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed
WO-1999030713-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed
WO-1999031061-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed
WO-1998046220-A1 COMBINATION THERAPY FOR THE PREVENTION AND TREATMENT OF OSTEOPOROSIS MERCK & CO., INC. (US) 1998-10-22 WO disclosed
WO-1998031359-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-07-23 WO disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed