SCHEMBL3870189

SCHEMBL3870189

O=C(NCCC(O)c1cccc(CC#CCC2CCCC2)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.35
OPRK1 P41145 3/20 0.34
OPRD1 P41143 2/20 0.34
MTNR1A P48039 3/20 0.33
MTNR1B P49286 3/20 0.33
GRIN2B Q13224 1/20 0.33
KLK7 P49862 1/20 0.32
CNR1 P21554 3/20 0.32
CNR2 P34972 3/20 0.32
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3865994 0.85 MTNR1A (0.40) OPRK1OPRD1MTNR1AMTNR1BCNR1
SCHEMBL3869016 0.82 CNR1 (0.36) OPRK1OPRD1MTNR1AMTNR1BCNR1
SCHEMBL3861226 0.81 MTNR1A (0.36) OPRK1OPRD1MTNR1AMTNR1BCNR1
SCHEMBL236172 0.80 MTNR1A (0.36) HDAC6OPRK1OPRD1MTNR1AMTNR1B
SCHEMBL235733 0.80 HDAC6 (0.36) HDAC6OPRK1OPRD1MTNR1AMTNR1B
SCHEMBL235732 0.80 HDAC6 (0.36) HDAC6OPRK1OPRD1MTNR1AMTNR1B
SCHEMBL13400259 0.76 HDAC6 (0.38) HDAC6OPRK1OPRD1MTNR1AMTNR1B
SCHEMBL2207058 0.76 SIRT2 (0.42)
SCHEMBL13400239 0.76 HDAC6 (0.38) HDAC6OPRK1OPRD1MTNR1AMTNR1B
SCHEMBL2207061 0.76 SIRT2 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed