SCHEMBL3870352

SCHEMBL3870352

CCn1cc(C(=O)OC2CC2)c(=O)c2c(N)c(F)c(F)c(F)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOXO1 Q12778 1/20 0.44
STAT3 P40763 1/20 0.43
HTT P42858 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
GSK3B P49841 5/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
CACNA1F O60840 1/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
CACNA1D Q01668 1/20 0.36
KCNH2 Q12809 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
TOP2A P11388 1/20 0.36
TOP2B Q02880 1/20 0.36
HTR3A P46098 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3870889 0.87 FOXO1 (0.40) FOXO1STAT3HTTKDM4EALDH1A1
SCHEMBL5868740 0.81 FOXO1 (0.53) FOXO1STAT3HTTKDM4EALDH1A1
SCHEMBL7158963 0.80 KDM4E (0.49) STAT3KDM4EALDH1A1TDP1HTR3A
SCHEMBL10723280 0.78 TDP1 (0.37) FOXO1STAT3HTTALDH1A1GSK3B
SCHEMBL3874174 0.78 FOXO1 (0.36) FOXO1STAT3HTTKDM4EALDH1A1
SCHEMBL27287068 0.76 STAT3 (0.70) STAT3HTTKDM4EALDH1A1CYP1A2
SCHEMBL1344898 0.76 STAT3 (0.54) STAT3HTTGSK3BCACNA1FPOLB
SCHEMBL3868260 0.75 GSK3B (0.42) FOXO1STAT3HTTKDM4EALDH1A1
SCHEMBL8111738 0.74 STAT3 (0.60) STAT3HTTKDM4EALDH1A1CYP1A2
SCHEMBL10857506 0.74 HPGD (0.44) STAT3KDM4EALDH1A1TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013182-A2 AMINOQUINOLONES AS GSK-3 INHIBITORS Activx Biosciences, Inc. (US) 2009-01-14 EP disclosed
WO-2007106537-A2 AMINOQUINOLONES AS GSK-3 INHIBITORS ACTIVX BIOSCIENCES, INC. (US) 2007-09-20 WO disclosed