SCHEMBL3873803

SCHEMBL3873803

Clc1ccc(C(c2ccc3nnn(Cc4ccccc4)c3c2)n2cncn2)cc1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.67
CYP11B1 P15538 1/20 0.67
TDP1 Q9NUW8 1/20 0.48
GRM2 Q14416 4/20 0.45
SLC9A1 P19634 1/20 0.45
CYP26A1 O43174 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3873165 0.95 CYP19A1 (0.71) CYP19A1CYP11B1TDP1GRM2
SCHEMBL3872062 0.91 CYP19A1 (0.66) CYP19A1CYP11B1TDP1CYP26A1KDM4E
SCHEMBL12189214 0.86 CYP19A1 (0.71) CYP19A1CYP11B1
SCHEMBL3879141 0.82 CYP19A1 (0.72) CYP19A1CYP11B1SLC9A1
SCHEMBL14092717 0.81 CYP19A1 (0.59) CYP19A1TDP1GRM2SLC9A1CYP26A1
SCHEMBL3872061 0.81 CYP19A1 (0.70) CYP19A1CYP11B1CYP26A1
SCHEMBL3871739 0.81 CYP19A1 (0.76) CYP19A1CYP11B1CYP26A1
Rac-Vorozole SCHEMBL13223107 0.80 CYP19A1 (1.00) CYP19A1CYP11B1
Vorozole SCHEMBL4554 0.80 CYP19A1 (1.00) CYP19A1CYP11B1
Rac-Vorozole SCHEMBL29606650 0.80 CYP19A1 (1.00) CYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874304-B1 BENZOTRIAZOLE DERIVATIVES AS CANNABINOID RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2009-07-15 EP claimed